BDBM469149 4-[6-(cyclopropylmethoxy)-1-methyl-3- methylsulfonylindazol-5-yl]-2- methylisoquinolin-1-one::US10807982, Example 29
SMILES Cn1nc(c2cc(c(OCC3CC3)cc12)-c1cn(C)c(=O)c2ccccc12)S(C)(=O)=O
InChI Key InChIKey=MSZYABAQZIIOQC-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469149
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair