BDBM469150 4-[6-(cyclopropylmethoxy)-3-ethylsulfonyl-1- methylindazol-5-yl]-2-methylisoquinolin-1-one::US10807982, Example 30
SMILES CCS(=O)(=O)c1nn(C)c2cc(OCC3CC3)c(cc12)-c1cn(C)c(=O)c2ccccc12
InChI Key InChIKey=AWTVHDWTTKQFKP-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469150
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair