BDBM469156 N-[6-(1,5-dimethyl-6-oxopyridin-3-yl)-1-[(3- fluorophenyl)methyl]-2-methylbenzimidazol-4- yl]ethanesulfonamide::US10807982, Example 36
SMILES CCS(=O)(=O)Nc1cc(cc2n(Cc3cccc(F)c3)c(C)nc12)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=CRGKRTPUIKQWDP-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469156
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair