BDBM469166 N-[6-(1,5-dimethyl-6-oxopyridin-3-yl)-1-[(2R)-1- methoxypropan-2-yl]-2-methylbenzimidazol-4- yl]methanesulfonamide::US10807982, Example 46
SMILES COC[C@@H](C)n1c(C)nc2c(NS(C)(=O)=O)cc(cc12)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=NRNTWQJZJADSJD-CYBMUJFWSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469166
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair