BDBM469168 N-[2-cyclopropyl-7-(2-methyl-1-oxoisoquinolin- 4-yl)-1,3-benzoxazol-5-yl]ethanesulfonamide::US10807982, Example 48
SMILES CCS(=O)(=O)Nc1cc(-c2cn(C)c(=O)c3ccccc23)c2oc(nc2c1)C1CC1
InChI Key InChIKey=QOFZCQYGEZDEJL-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469168
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair