BDBM469169 4-[7-(cyclopropylmethoxy)-4-ethylsulfonyl-2,3- dihydro-1,4-benzoxazin-6-yl]-2- methylisoquinolin-1-one::US10807982, Example 49
SMILES CCS(=O)(=O)N1CCOc2cc(OCC3CC3)c(cc12)-c1cn(C)c(=O)c2ccccc12
InChI Key InChIKey=PVWHOYFZJDGCRS-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469169
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair