BDBM469171 N-[2-cyclopropyl-7-(1,5-dimethyl-6-oxopyridin- 3-yl)-1,3-benzoxazol-5-yl]propane-2-sulfonamide::US10807982, Example 51
SMILES CC(C)S(=O)(=O)Nc1cc(-c2cc(C)c(=O)n(C)c2)c2oc(nc2c1)C1CC1
InChI Key InChIKey=ASJMQONOWHRNLT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469171
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair