BDBM469172 N-[2-cyclopropyl-7-(1,5-dimethyl-6-oxopyridin-3- yl)-1,3-benzoxazol-5-yl]ethanesulfonamide::US10807982, Example 52
SMILES CCS(=O)(=O)Nc1cc(-c2cc(C)c(=O)n(C)c2)c2oc(nc2c1)C1CCCC1
InChI Key InChIKey=YOMMCHWWGKGIIB-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469172
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair