BDBM469173 N-[2-cyclopentyl-7-(2-methyl-1-oxoisoquinolin-4- yl)-1,3-benzoxazol-5-yl]ethanesulfonamide::US10807982, Example 53
SMILES CCS(=O)(=O)Nc1cc(-c2cn(C)c(=O)c3ccccc23)c2oc(nc2c1)C1CCCC1
InChI Key InChIKey=VUNICRAJLKWEQG-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469173
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair