BDBM469175 N-[2-cyclopropyl-3-methyl-7-(2-methyl-1- oxoisoquinolin-4-yl)benzimidazol-5- yl]ethanesulfonamide::US10807982, Example 55
SMILES CCS(=O)(=O)Nc1cc(-c2cn(C)c(=O)c3ccccc23)c2nc(C3CC3)n(C)c2c1
InChI Key InChIKey=USCXTHQXBKFRGG-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469175
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair