BDBM469177 N-[2-cyclopentyl-7-(5-methoxy-1-methyl-6- oxopyridin-3-yl)-1,3-benzoxazol-5- yl]ethanesulfonamide::US10807982, Example 57
SMILES CCS(=O)(=O)Nc1cc(-c2cc(OC)c(=O)n(C)c2)c2oc(nc2c1)C1CCCC1
InChI Key InChIKey=TYHDAJBFQXYGBK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469177
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair