BDBM469179 5-[6-(cyclopropylmethoxy)-1-methyl-3- methylsulfonylindazol-5-yl]-3-methoxy-1- methylpyridin-2-one::US10807982, Example 59
SMILES COc1cc(cn(C)c1=O)-c1cc2c(cc1OCC1CC1)N(C)N=S2S(C)(=O)=O
InChI Key InChIKey=MXLVVBOODMBVOJ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469179
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair