BDBM469182 N-[1-[(2,4-difluorophenyl)methyl]-6-(1,5- dimethyl-6-oxopyridin-3-yl)-2- methylimidazo[4,5-c]pyridin-4- yl]methanesulfonamide::US10807982, Example 62
SMILES Cc1nc2c(NS(C)(=O)=O)nc(cc2n1Cc1ccc(F)cc1F)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=TXHGJPUHHSRHLZ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469182
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair