BDBM469185 N-[3-fluoro-1-[(4-fluorophenyl)methyl]-6-(5- methoxy-1-methyl-6-oxopyridin-3-yl)indazol-4- yl]methanesulfonamide::US10807982, Example 65
SMILES COc1cc(cn(C)c1=O)-c1cc(NS(C)(=O)=O)c2c(F)nn(Cc3ccc(F)cc3)c2c1
InChI Key InChIKey=OEFLTDFHTBWWIW-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469185
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair