BDBM469190 5-[3-(cyclopropylmethyl)-7-ethylsulfonyl-2- methylbenzimidazol-5-yl]-3-methoxy-1- methylpyridin-2-one::US10807982, Example 70
SMILES CCS(=O)(=O)c1cc(cc2n(CC3CC3)c(C)nc12)-c1cc(OC)c(=O)n(C)c1
InChI Key InChIKey=OMLUYJWWXPMJJZ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469190
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair