BDBM469195 5-(1-ethyl-4-methylsulfonylindol-2-yl)-1,3- dimethylpyridin-2-one::US10807982, Example 75
SMILES CCn1c(cc2c(cccc12)S(C)(=O)=O)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=HITUUJQTXLWNJZ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469195
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair