BDBM469197 4-[1-(cyclopropylmethyl)-4-methylsulfonylindol- 2-yl]-2-methylisoquinolin-1-one::US10807982, Example 78
SMILES Cn1cc(-c2cc3c(cccc3n2CC2CC2)S(C)(=O)=O)c2ccccc2c1=O
InChI Key InChIKey=PPIGOOJJBPANIV-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469197
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair