BDBM469199 N-[2-cyclopropyl-7-(1,5-dimethyl-6-oxopyridin- 3-yl)-1-benzofuran-5-yl]methanesulfonamide::US10807982, Example 80
SMILES Cc1cc(cn(C)c1=O)-c1cc(NS(C)(=O)=O)cc2cc(oc12)C1CC1
InChI Key InChIKey=LHEMTKPEUZEKNE-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469199
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair