BDBM469210 5-[1-(2-cyclopropylethyl)-4-methylsulfonylindol- 2-yl]-3-methoxy-1-methylpyridin-2-one::US10807982, Example 91
SMILES COc1cc(cn(C)c1=O)-c1cc2c(cccc2n1CCC1CC1)S(C)(=O)=O
InChI Key InChIKey=BCDGLJJQDDUILV-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469210
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair