BDBM469212 N-[1-(cyclopropylmethyl)-6-(5-methoxy-1- methyl-6-oxopyridin-3-yl)-2- (trifluoromethyl)benzimidazol-4- yl]methanesulfonamide::US10807982, Example 93
SMILES COc1cc(cn(C)c1=O)-c1cc(NS(C)(=O)=O)c2nc(n(CC3CC3)c2c1)C(F)(F)F
InChI Key InChIKey=UGRKFNYEYMCTHS-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469212
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair