BDBM469216 5-[3-(cyclopropylmethyl)-2-ethoxy-7- (methylsulfonylmethyl)benzimidazol-5-yl]-1,3- dimethylpyridin-2-one::US10807982, Example 97
SMILES CCOc1nc2c(CS(C)(=O)=O)cc(cc2n1CC1CC1)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=QHKMXVMYKLXAGR-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469216
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair