BDBM469219 5-[2-cyclopropyl-5-(ethylsulfonylmethyl)-1,3- benzoxazol-7-yl]-3-methoxy-1- methylpyridin-2-one::US10807982, Example 100
SMILES CCS(=O)(=O)Cc1cc(-c2cc(OC)c(=O)n(C)c2)c2oc(nc2c1)C1CC1
InChI Key InChIKey=ITDJQMDKFBKZOG-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469219
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair