BDBM469224 N-[6-(1,5-dimethyl-6-oxopyridin-3-yl)-3-fluoro-1- [(4-fluorophenyl)methyl]indazol-4- yl]ethanesulfonamide::US10807982, Example 105
SMILES CCS(=O)(=O)Nc1cc(cc2n(Cc3ccc(F)cc3)nc(F)c12)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=LCPICCSRZFYNOI-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 469224
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BREM was cloned, expr...More data for this Ligand-Target Pair