BDBM475412 1-[5-(3-Hydroxy-phenyl)-1H-benzoimidazol-2-yl]-1H-::US10851083, Example 24::US11618744, Example 24

SMILES OC(=O)c1cnn(c1)-c1nc2cc(ccc2[nH]1)-c1cccc(O)c1

InChI Key InChIKey=LZXBZILJESOINQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 475412   

TargetEgl nine homolog 1 [181-417](Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM475412(1-[5-(3-Hydroxy-phenyl)-1H-benzoimidazol-2-yl]-1H-...)
Affinity DataIC50:  316nMAssay Description:The PHD2 181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypep...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEgl nine homolog 1 [181-417](Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM475412(1-[5-(3-Hydroxy-phenyl)-1H-benzoimidazol-2-yl]-1H-...)
Affinity DataIC50:  316nMAssay Description:The PHD2181-417 polypeptide (3 μg) was pre-incubated for 30 minutes with test compound prior to assessing the enzymatic activity of the polypept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent