BDBM475690 (4aS*,8aR*)-2- (5-bromo-4- methyl-2- pyridyl)-8a- methyl-7-(7H- pyrrolo[2,3- d]pyrimidin-4- yl)- 3,4,4a,5,6,8- hexahydro-1H- 2,7- naphthyridine::US10851116, Example 12
SMILES Cc1cc(ncc1Br)N1CC[C@H]2CCN(C[C@@]2(C)C1)c1ncnc2[nH]ccc12
InChI Key
Data 4 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 475690
Affinity DataEC50: 203nMAssay Description:Inhibition of phosphorylation of a synthetic peptide was measured in an HTRF-based assay using the TK substrate-Biotin from the Cisbio HTRFKinEASE TK...More data for this Ligand-Target Pair
Affinity DataEC50: 4.27E+3nMAssay Description:Inhibition of phosphorylation of a synthetic peptide was measured in an HTRF-based assay using the TK substrate-Biotin from the Cisbio HTRFKinEASE TK...More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Inhibition of phosphorylation of a synthetic peptide was measured in an HTRF-based assay using the TK substrate-Biotin from the Cisbio HTRFKinEASE TK...More data for this Ligand-Target Pair
Affinity DataEC50: 937nMAssay Description:Inhibition of phosphorylation of a synthetic peptide was measured in an HTRF-based assay using the TK substrate-Biotin from the Cisbio HTRFKinEASE TK...More data for this Ligand-Target Pair