BDBM476471 (2S)-4-[(4S,5S)-5-(2-cyanophenyl)-4- methyl-4,5-dihydro-1,3-oxazol-2-yl]- 1-[N2-cyclohexyl-N6-(methylsulfonyl)- D-lysyl]-N-(thiophen-2- ylmethyl)piperazine-2-carboxamide::US10875851, Example 127
SMILES C[C@@H]1N=C(O[C@H]1c1ccccc1C#N)N1CCN([C@@H](C1)C(=O)NCc1cccs1)C(=O)[C@@H](CCCCNS(C)(=O)=O)NC1CCCCC1
InChI Key InChIKey=UBEIAGOISNYVQV-QIXIFPRPSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 476471
Affinity DataIC50: 18.7nMAssay Description:The effectiveness of a compound of the present invention as an inhibitor of Coagulation Factor XIIa can be determined using a relevant purified serin...More data for this Ligand-Target Pair