BDBM477646 US10889568, Compound 21::[4-(6-Amino-5-methoxy-pyridazin-3- yl)-piperidin-1-yl]-(4-methoxy-5- phenoxy-pyridin-2-yl)-methanone

SMILES COc1cc(nnc1C)C1CCN(CC1)C(=O)c1cc(OC)c(Oc2ccccc2)cn1

InChI Key InChIKey=GNKYCOIDYFVTDZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 477646   

TargetShort transient receptor potential channel 6(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM477646(US10889568, Compound 21 | [4-(6-Amino-5-methoxy-py...)
Affinity DataIC50:  43nMAssay Description:The commercially available HEK293/TREx line (Invitrogen) was stably transfected with a TRPC6 construct and screened by conventional calcium imaging t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent