BDBM477652 US10889568, Compound 27::[(R)-4-(6-Amino-4-methoxy-pyridin- 3-yl)-2-methoxymethyl-piperazin-1- yl]-(4-methoxy-5-phenoxy-pyridin-2- yl)-methanone

SMILES COC[C@H]1CN(CCN1C(=O)c1cc(OC)c(Oc2ccccc2)cn1)c1cnc(C)cc1OC

InChI Key InChIKey=MJHSCZLPVWNOPZ-LJQANCHMSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 477652   

TargetShort transient receptor potential channel 6(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM477652(US10889568, Compound 27 | [(R)-4-(6-Amino-4-methox...)
Affinity DataIC50:  75nMAssay Description:The commercially available HEK293/TREx line (Invitrogen) was stably transfected with a TRPC6 construct and screened by conventional calcium imaging t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent