BDBM483874 N-methyl-1-(cis-5- (methyl(2- (trifluoromethyl)- benzyl)amino)- octahydrocyclopenta- [c]pyrrole-2- carbonyl)-1H- pyrazole-3- carboxamide::US10927105, Ex 434::US11655217, Example 434

SMILES CNC(=O)c1ccn(n1)C(=O)N1C[C@@H]2C[C@@H](C[C@@H]2C1)N(C)Cc1ccccc1C(F)(F)F

InChI Key InChIKey=DSIIGPMACNPLQG-BJWYYQGGSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 483874   

TargetMonoglyceride lipase(Homo sapiens (Human))
H. Lundbeck

US Patent
LigandPNGBDBM483874(N-methyl-1-(cis-5- (methyl(2- (trifluoromethyl)- b...)
Affinity DataIC50: <100nMAssay Description:Proteomes (mouse brain membrane fraction for mouse assays; human prefrontal cortex membrane fractions for human assays) (50 mL, 1.0 mg/mL total prote...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMonoglyceride lipase(Homo sapiens (Human))
H. Lundbeck

US Patent
LigandPNGBDBM483874(N-methyl-1-(cis-5- (methyl(2- (trifluoromethyl)- b...)
Affinity DataIC50: <100nMAssay Description:Proteomes (mouse brain membrane fraction for mouse assays; human prefrontal cortex membrane fractions for human assays) (50 mL, 1.0 mg/mL total prote...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent