BDBM48532 2-butoxy-N-[2-(diethylamino)ethyl]-4-quinolinecarboxamide;hydrochloride::2-butoxy-N-[2-(diethylamino)ethyl]cinchoninamide;hydrochloride::2-butoxy-N-[2-(diethylamino)ethyl]quinoline-4-carboxamide;hydrochloride::Cincain::Cinchocaine::DIBUCAINE HYDROCHLORIDE::Dibucaine::MLS000028429::Nupercainal::Nupercaine::SMR000058369::Sovcaine::cid_521951

SMILES CCCCOc1cc(C(=O)NCCN(CC)CC)c2ccccc2n1

InChI Key InChIKey=PUFQVTATUTYEAL-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 48532   

TargetEukaryotic translation initiation factor 4 gamma 1(Homo sapiens (Human))
Emory University

Curated by PubChem BioAssay
LigandPNGBDBM48532(2-butoxy-N-[2-(diethylamino)ethyl]-4-quinolinecarb...)
Affinity DataIC50:  5.00E+4nMAssay Description:Dose Response Confirmation for Small Molecule Inhibitors of Eukaryotic Translation Initiation NIH Molecular Libraries Screening Centers Network [MLSC...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetBile salt export pump(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM48532(2-butoxy-N-[2-(diethylamino)ethyl]-4-quinolinecarb...)
Affinity DataIC50:  4.17E+4nMAssay Description:Ability to inhibit HMG-CoA reductase (HMGR) by CoA reductase inhibition screen (COR) in ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM48532(2-butoxy-N-[2-(diethylamino)ethyl]-4-quinolinecarb...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of binding of Batrachotoxinin [3H]BTX-B to high affinity sites on voltage dependent sodium channels in a vesicular preparation from guinea...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed