BDBM485745 3-(isoquinolin-5-yloxy)- N,N-dimethyl-3-(thiophen- 2-yl)propan-1-amine::US10941138, Example 43
SMILES CN(C)CCC(Oc1cccc2cnccc12)c1cccs1
InChI Key InChIKey=MRFWCXUEQACNJT-UHFFFAOYSA-N
Data 1 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 485745
TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Homo sapiens (Human))
Esteve Pharmaceuticals
US Patent
Esteve Pharmaceuticals
US Patent
Affinity DataKi: 1.75E+3nMAssay Description:Human α2δ-1 enriched membranes (2.5 μg) were incubated with 15 nM of radiolabeled [3H]-Gabapentin in assay buffer containing Hepes-KOH...More data for this Ligand-Target Pair