BDBM486384 3-(3-cyclopropylphenyl)-N-(1,1- dioxidotetrahydrothiophen-3-yl)-1-(5- fluoropyrimidin-2-yl)-1H-indole-6- carboxamide (enantiomer A)::US10947222, Example 17-A
SMILES Fc1cnc(nc1)-n1cc(-c2cccc(c2)C2CC2)c2ccc(cc12)C(=O)N[C@H]1CCS(=O)(=O)C1
InChI Key InChIKey=YHDGYDULNRWBKV-NRFANRHFSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 486384
Affinity DataIC50: 3.30nMAssay Description:DGAT2 activity was determined by measuring the amount of enzymatic product triolein (1,2,3-Tri(cis-9-octadecenoyl)glycerol) using the membrane prep m...More data for this Ligand-Target Pair