BDBM486547 US10947251, Example 24
SMILES Fc1cc(N2[C@H]3CCN(C[C@@H]3OCC2=O)S(=O)(=O)Nc2ccon2)c(cc1-c1cccc(c1)C(F)(F)F)C#N
InChI Key InChIKey=BMPKQQGNTVQMHQ-FPOVZHCZSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 486547
Affinity DataIC50: 237nMAssay Description:Patch voltage clamp electrophysiology allows for the direct measurement and quantification of block of voltage-gated sodium channels (NaV's), and...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Heterologously Express hNav1.7 and the β1 SubunitPreparation of membranes containing recombinantly expressed sodium channels: Frozen recombinant...More data for this Ligand-Target Pair