BDBM50010696 (R)-2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol::2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinoline-10,11-diol::CHEMBL276326

SMILES CN1CCc2cc(Br)cc-3c2[C@H]1Cc1ccc(O)c(O)c-31

InChI Key InChIKey=SETZXJXEHHDPBP-CYBMUJFWSA-N

Data  3 KI  2 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50010696   

TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50010696((R)-2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenz...)
Affinity DataKi:  17.7nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50010696((R)-2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenz...)
Affinity DataKi:  18nMAssay Description:Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50010696((R)-2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenz...)
Affinity DataKi:  106nMAssay Description:Binding affinity at rat striatal Dopamine receptor D1 using [3H]- SCH-23390 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50010696((R)-2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenz...)
Affinity DataKd:  728nMAssay Description:Compound was evaluated for the ability to displace [3H]-spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as low affinity stateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50010696((R)-2-Bromo-6-methyl-5,6,6a,7-tetrahydro-4H-dibenz...)
Affinity DataKd:  6.80nMAssay Description:Compound was evaluated for the ability to displace [3H]-spiperone at Dopamine receptor D2 in porcine anterior pituitary gland as high affinity stateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed