BDBM50094894 CHEMBL3589485

SMILES O=C(N1CC(=O)Nc2ccccc12)c1cncc(c1)-c1ccccc1

InChI Key InChIKey=LRMDXTVKVHKWEK-UHFFFAOYSA-N

Data  2 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50094894   

TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094894(CHEMBL3589485)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094894(CHEMBL3589485)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed