BDBM50206038 ((2S,4S)-4-(4-(4-nitrophenyl)piperazin-1-yl)pyrrolidin-2-yl)(thiazolidin-3-yl)methanone::CHEMBL391466
SMILES [O-][N+](=O)c1ccc(cc1)N1CCN(CC1)[C@@H]1CN[C@@H](C1)C(=O)N1CCSC1
InChI Key InChIKey=ZHJLERMYNKCYGH-IRXDYDNUSA-N
Data 8 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50206038
Affinity DataIC50: 2.20nMAssay Description:Inhibition of DPP4 in rat plasma by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-MCA as substrate after 60 mins by fluorometryMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human DPP9 using GLY-Pro-MCA as substrate after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30.2nMAssay Description:Inhibition of human recombinant DPP9 using Gly-Pro-MCA as substrate after 30 mins by fluorometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of DPP4 in human plasma using GLY-Pro-MCA as substrate after 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human DPP8 using GLY-Pro-MCA as substrate after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12.2nMAssay Description:Inhibition of human recombinant DPP8 using Gly-Pro-MCA as substrate after 30 mins by fluorometryMore data for this Ligand-Target Pair