BDBM50273099 3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[c]pyrazole::3-(2H-tetrazol-5-yl)-1,4,5,6-tetrahydro-cyclopentapyrazole::CHEMBL456145::MK-0354
SMILES C1Cc2[nH]nc(c2C1)-c1nnn[nH]1
InChI Key InChIKey=LTQYSJKGRPGMPO-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50273099
Affinity DataKi: 505nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.08E+3nMAssay Description:Agonist activity against mouse GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity against human GPR109a assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity against mouse GPR109a assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity against rat GPR109a assessed as GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 286nMAssay Description:Agonist activity at human GPR109a expressed in CHO cells assessed as decrease in forskolin-stimulated cAMP production by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.65E+3nMAssay Description:Agonist activity against human GPR109a assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR10a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR10a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 286nMAssay Description:Agonist activity at GPR109a expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production by HTRF assayMore data for this Ligand-Target Pair