BDBM50426501 CHEMBL2323578

SMILES CCNC(=O)N(CCCN1CCOCC1)C(=O)[C@@H]1C[C@H]2[C@@H](Cc3c[nH]c4cccc2c34)N(CC=C)C1

InChI Key InChIKey=GIVLQJIZLYGZTG-GZGNHOFSSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50426501   

Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50426501(CHEMBL2323578)
Affinity DataKi:  7.10nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50426501(CHEMBL2323578)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human 5-HT2B receptor transfected in CHO cell assessed as IP1 production incubated for 30 mins measured by HTRF detection methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed