BDBM50444496 CHEMBL3092650
SMILES O=C1CCCN1c1ccc(Oc2ccc3CCN(CCc3c2)C2CCC2)nc1
InChI Key InChIKey=YFRBKEVUUCQYOW-UHFFFAOYSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50444496
Affinity DataKi: 0.148nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from rat histamine H3 receptor expressed in HEK293 cells after 45 mins by liquid scintillation spectromet...More data for this Ligand-Target Pair
Affinity DataKi: 0.363nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+3nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >3.16E+3nMAssay Description:Binding affinity to human histamine H2 receptorMore data for this Ligand-Target Pair