BDBM50445253 CHEMBL1232500

SMILES CCN1C(Sc2ccc(O)cc12)=CC(C)=O

InChI Key InChIKey=GCSZJMUFYOAHFY-UHFFFAOYSA-N

Data  3 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50445253   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50445253(CHEMBL1232500)
Affinity DataIC50:  240nMAssay Description:Inhibition of Dyrk1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50445253(CHEMBL1232500)
Affinity DataIC50:  240nMAssay Description:Inhibition of human recombinant full length GST-tagged DYRK1A expressed in baculovirus expression system after 10 mins in presence of [gamma33P-ATP] ...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)

Curated by ChEMBL
LigandPNGBDBM50445253(CHEMBL1232500)
Affinity DataIC50:  240nMAssay Description:Competitive inhibition of DYRK1A (unknown origin) using ATPMore data for this Ligand-Target Pair