BDBM50503685 CHEMBL4092241
SMILES [H][C@]12CN3CC(=C1)[C@]1([H])CCN(C[C@@]1([H])CC\C=C/CCCC3)CCCC\C=C/CC2
InChI Key InChIKey=UOAQLFVPXKOHCQ-ZUCXHZAFSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50503685
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of 20s constitutive proteasome beta2 trypsin-like activity in human erythrocytes using Boc-Leu-Arg-Arg-MCA as substrate preincubated for 1...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of 20s immunoproteasome LMP2 in human erythrocytes using Ac-Pro-Ala-Leu-MCA as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of 20s immunoproteasome MECL1 in human erythrocytes using Suc-Leu-Leu-ValTyr-MCA as substrate preincubated for 10 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of 20s constitutive proteasome beta5 chymotrypsin-like activity in human erythrocytes using Suc-Leu-Leu-ValTyr-MCA as substrate preincubat...More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of 20s constitutive proteasome beta1 caspase-like activity in human erythrocytes using Boc-Leu-Arg-Arg-MCA as substrate preincubated for 1...More data for this Ligand-Target Pair
Affinity DataIC50: 630nMAssay Description:Inhibition of 20s immunoproteasome LMP7 in human erythrocytes using Suc-Leu-Leu-ValTyr-MCA as substrate preincubated for 10 mins followed by substrat...More data for this Ligand-Target Pair