BDBM50515599 CHEMBL4457426
SMILES COc1cc(\C=C\C(=O)NCCN2CCC(CCC(=O)c3cc(Cl)c(N)cc3OC)CC2)ccc1O
InChI Key InChIKey=GRSPTEBOWFGVCL-VMPITWQZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50515599
Affinity DataKi: 101nMAssay Description:Binding affinity to recombinant human brain 5HT4 receptor by radio ligand binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Partial agonist activity at human HA-tagged 5HT4 receptor expressed in COS7 cells assessed as induction of cAMP production measured after 10 mins by ...More data for this Ligand-Target Pair
Affinity DataIC50: 101nMAssay Description:Displacement of [3H]-GR 113808 from recombinant human brain 5HT4 receptor measured after 60 mins by radio ligand binding assayMore data for this Ligand-Target Pair