BDBM75207 2-(5-bromanylthiophen-2-yl)-N-(3-ethoxypropyl)quinoline-4-carboxamide::2-(5-bromo-2-thienyl)-N-(3-ethoxypropyl)cinchoninamide::2-(5-bromo-2-thiophenyl)-N-(3-ethoxypropyl)-4-quinolinecarboxamide::2-(5-bromothien-2-yl)-N-(3-ethoxypropyl)quinoline-4-carboxamide::2-(5-bromothiophen-2-yl)-N-(3-ethoxypropyl)quinoline-4-carboxamide::MLS001197915::SMR000559708::cid_15996111

SMILES CCOCCCNC(=O)c1cc(nc2ccccc12)-c1ccc(Br)s1

InChI Key InChIKey=DNBQQPVZBPPQSW-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 75207   

TargetImportin subunit alpha-1(Homo sapiens (Human))
Broad Institute

Curated by PubChem BioAssay
LigandPNGBDBM75207(2-(5-bromanylthiophen-2-yl)-N-(3-ethoxypropyl)quin...)
Affinity DataEC50:  2.79E+4nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPhotoreceptor-specific nuclear receptor(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM75207(2-(5-bromanylthiophen-2-yl)-N-(3-ethoxypropyl)quin...)
Affinity DataIC50:  6.67E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Affiliation: The Scripps Research Institute, TSRI Assay Provide...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetIsoform 2 of Nuclear receptor corepressor 2 (TRAC-1)(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM75207(2-(5-bromanylthiophen-2-yl)-N-(3-ethoxypropyl)quin...)
Affinity DataIC50:  4.18E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center Affiliation: The Scripps Research Institute, TSRI Assay Provide...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay