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Found 18 Enz. Inhib. hit(s) with Target = '40S ribosomal protein S27'
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420401(CHEMBL2089255 | US11208696, Example 31)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of Mps1-mediated p38 MAPK phosphorylation after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420400(CHEMBL2089254)
Affinity DataIC50:  37nMAssay Description:Inhibition of Mps1-mediated p38 MAPK phosphorylation after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420401(CHEMBL2089255 | US11208696, Example 31)
Affinity DataIC50:  131nMAssay Description:Inhibition of FLAG-tagged Mps1 autophosphorylation in human RERF-LC-AI cells expressing Tet-suppressible promotor after 3 hrs by immunoblottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420399(CHEMBL2089253)
Affinity DataIC50:  228nMAssay Description:Inhibition of Mps1-mediated p38 MAPK phosphorylation after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM15912(2-pyridinecarboxamide deriv. 8b | 4-Amino-5-cyano-...)
Affinity DataIC50:  529nMAssay Description:Inhibition of Mps1-mediated p38 MAPK phosphorylation after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM15913(2-pyridinecarboxamide deriv. 8c | 4-Amino-5-cyano-...)
Affinity DataIC50:  568nMAssay Description:Inhibition of Mps1-mediated p38 MAPK phosphorylation after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420400(CHEMBL2089254)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of FLAG-tagged Mps1 autophosphorylation in human RERF-LC-AI cells expressing Tet-suppressible promotor after 3 hrs by immunoblottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420398(CHEMBL2089252)
Affinity DataIC50:  3.97E+3nMAssay Description:Inhibition of Mps1-mediated p38 MAPK phosphorylation after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM15926(Aminopyridine-Based Inhibitor 6e | N-(4-Amino-5-cy...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of Mps1-mediated p38 MAPK phosphorylation after 90 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50361088(CHEMBL1933582)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50361089(CHEMBL1933576)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048374(CHEMBL3310151)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048365(CHEMBL3309998)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048364(CHEMBL3309997)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048362(CHEMBL3309995)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50048357(CHEMBL3309990)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021626(CHEMBL3298400)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target40S ribosomal protein S27(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021618(CHEMBL3297762 | US9145418, 2)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MPS1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed