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Found 15 Enz. Inhib. hit(s) with Target = 'Guanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2'
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230850(US9346793, 1)
Affinity DataEC50:  11.8nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230864(US9346793, 15)
Affinity DataEC50:  52.9nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230852(US9346793, 3)
Affinity DataEC50:  8nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230853(US9346793, 4)
Affinity DataEC50:  51nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230854(US9346793, 5)
Affinity DataEC50:  21.7nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230855(US9346793, 6)
Affinity DataEC50:  12.7nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230856(US9346793, 7)
Affinity DataEC50:  10.1nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230857(US9346793, 8)
Affinity DataEC50:  17.8nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230858(US9346793, 9)
Affinity DataEC50:  17.2nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230859(US9346793, 10)
Affinity DataEC50:  10.3nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230860(US9346793, 11)
Affinity DataEC50:  82.3nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230861(US9346793, 12)
Affinity DataEC50:  32.3nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230862(US9346793, 13)
Affinity DataEC50:  13.2nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230863(US9346793, 14)
Affinity DataEC50:  11.3nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGuanine nucleotide-binding protein subunit alpha-15 [Y147C]/N-formyl peptide receptor 2(Homo sapiens (Human))
Actelion Pharmaceuticals

US Patent
LigandPNGBDBM230851(US9346793, 2)
Affinity DataEC50:  7.60nMAssay Description:Cells expressing recombinant human ALX receptor and the G-protein Gα16 (HEK293-hALXR-Gα16) were grown to 80% confluency in Growing Medium (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent