TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 4.56E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 7.87E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 7.87E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 9.64E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.21E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) at pH ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.65E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.99E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.03E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 2.70E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: >3.33E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 H381R mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 5.13E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.04E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.07E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 1.14E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 2.56E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.19E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.22E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.24E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.39E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 M424A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.43E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.72E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.83E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.85E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 3.93E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 4.62E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataIC50: 5.35E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 M424A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibitory activity towards Beta-Glucosidase from Caldocellum saccharolMore data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 280nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 2.60E+4nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of T effector cells mediated K562 cell lysis preincubated with K562 cells ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 1.60nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of T effector cells mediated K562 cell lysis preincubated with K562 cells ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 4.10E+4nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of T effector cells mediated K562 cell lysis preincubated with K562 cells ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 7.30E+3nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of T effector cells mediated K562 cell lysis preincubated with K562 cells ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataKd: 1.11E+5nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 5.40nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 4.00E+3nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 0.510nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 8.90nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 0.0600nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 487nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 1.40nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University
Curated by ChEMBL
Western Michigan University
Curated by ChEMBL
Affinity DataEC50: 0.450nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair