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Found 151 Enz. Inhib. hit(s) with Target = 'Butyrophilin subfamily 3 member A1'
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  4.56E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516697(CHEMBL4302450)
Affinity DataIC50:  7.87E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516697(CHEMBL4302450)
Affinity DataIC50:  7.87E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  9.64E+3nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.21E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) at pH ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.61E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.65E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  1.99E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50:  2.30E+4nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516698(CHEMBL4116247)
Affinity DataIC50:  1.03E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516699(CHEBI:16057 | DIMETHYLALLYL DIPHOSPHATE | Dimethyl...)
Affinity DataIC50:  2.70E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataIC50: >3.33E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 H381R mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM25257(({hydroxy[(3-methylbut-3-en-1-yl)oxy]phosphoryl}ox...)
Affinity DataIC50:  5.13E+5nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  1.04E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  1.07E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50278316(CHEMBL450079 | sodium pyrophosphate(V))
Affinity DataIC50:  1.14E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  2.56E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 B30.2 domain (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.19E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.22E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.24E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 W421A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.39E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 M424A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.43E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R442A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  3.72E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.83E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R499A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.85E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 full interaction domain (unknown origin) expressed in Escherichia coli BL21 (DE) measur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataIC50:  3.93E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  4.62E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 R448A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50516696(CHEMBL4521062)
Affinity DataIC50:  5.35E+6nMAssay Description:Displacement of GDP-BODIPY from C-terminal 6His-tagged BTN3A1 M424A mutant (unknown origin) expressed in Escherichia coli BL21 (DE) measured after 60...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236888(CHEMBL4097373)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibitory activity towards Beta-Glucosidase from Caldocellum saccharolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236889(CHEMBL4061531)
Affinity DataEC50:  41nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236888(CHEMBL4097373)
Affinity DataEC50: >1.00E+5nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236889(CHEMBL4061531)
Affinity DataEC50:  280nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236890(CHEMBL4089656)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236891(CHEMBL4081059)
Affinity DataEC50: >1.00E+5nMAssay Description:Displacement of [3H]spiperone from human Dopamine receptor D3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236892(CHEMBL4099094)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of T effector cells mediated K562 cell lysis preincubated with K562 cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataEC50:  1.60nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of T effector cells mediated K562 cell lysis preincubated with K562 cells ...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236890(CHEMBL4089656)
Affinity DataEC50:  4.10E+4nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of T effector cells mediated K562 cell lysis preincubated with K562 cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236891(CHEMBL4081059)
Affinity DataEC50:  7.30E+3nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of T effector cells mediated K562 cell lysis preincubated with K562 cells ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236892(CHEMBL4099094)
Affinity DataEC50: >1.00E+5nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataKd:  1.11E+5nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236895(CHEMBL4088948)
Affinity DataEC50:  5.40nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236894(CHEMBL4060737)
Affinity DataEC50:  4.00E+3nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataEC50:  0.510nMAssay Description:Activation of BTN3A1 in human Vgamma9Vdelta2 T cells assessed as induction of interleukin 2 stimulated cell proliferation treated for 72 hrs measured...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50271365(CHEMBL4127261)
Affinity DataEC50:  8.90nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50236893(CHEBI:15664 | CHEMBL145233)
Affinity DataEC50:  0.0600nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM12578(2-(imidazol-1-yl)-1-hydroxyethylidene-1,1-bisphosp...)
Affinity DataEC50:  487nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50271366(CHEMBL4126163)
Affinity DataEC50:  1.40nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetButyrophilin subfamily 3 member A1(Homo sapiens (Human))
Western Michigan University

Curated by ChEMBL
LigandPNGBDBM50271368(CHEMBL4126016)
Affinity DataEC50:  0.450nMAssay Description:Binding affinity to butyrophilin 3A1 in human Vgamma9/Vdelta2 T-cells assessed as activation of Vgamma9/Vdelta2 T-cells by upregulation of CD69 and C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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