Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with Target = 'Calcium-dependent protein kinase 4'
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM79181(10-[3-(4-methyl-1-piperazinyl)propyl]-2-(trifluoro...)
Affinity DataKi:  1.50E+5nMAssay Description:Inhibition of Plasmodium falciparum His-tagged CDPK4 expressed in Escherichia coli BL21(DE3) using EGTA as substrate after 10 mins in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50383381(CHEMBL2030554 | CHEMBL2070050 | US10544104, Compou...)
Affinity DataIC50:  4nMAssay Description:Inhibition of CDPK4 in Plasmodium falciparum 3D7 microgametesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50383381(CHEMBL2030554 | CHEMBL2070050 | US10544104, Compou...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Plasmodium falciparum CDPK4 using syntide-2 as substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50389704(CHEMBL2070081 | US10544104, Compound 150 | US95180...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Plasmodium falciparum CDPK4 using syntide-2 as substrate by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50345704(1-(tert-butyl)-3-(naphthalen-2-yl)-1H-pyrazolo[3,4...)
Affinity DataIC50:  177nMAssay Description:Inhibition of CDPK4 in Plasmodium falciparum 3D7 microgametesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50530659(CHEMBL4461850)
Affinity DataKd:  60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50530637(CHEMBL4591417)
Affinity DataKd:  50nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50530659(CHEMBL4461850)
Affinity DataKd:  60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50530659(CHEMBL4461850)
Affinity DataKd:  60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50530637(CHEMBL4591417)
Affinity DataKd:  50nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50530659(CHEMBL4461850)
Affinity DataKd:  60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50530637(CHEMBL4591417)
Affinity DataKd:  50nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
TBA

Curated by ChEMBL
LigandPNGBDBM50530637(CHEMBL4591417)
Affinity DataKd:  50nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed