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Found 7 Enz. Inhib. hit(s) with Target = 'Kallikrein-2'
TargetKallikrein-2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50396163(CHEMBL2171880)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of human KLK2 after 1 hr by phage-display based Immunofluorometric AssayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataKi:  1.60E+3nMAssay Description:Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50256262(CHEMBL4070056)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal 10His-tagged KLK2 (1 to 261 residues) expressed in mouse NS0 cells using fluorogenic PFR-AMC peptide as su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50256260(CHEMBL4094403)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of recombinant human C-terminal 10His-tagged KLK2 (1 to 261 residues) expressed in mouse NS0 cells using fluorogenic PFR-AMC peptide as su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50256261(CHEMBL4059991)
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of platelet-derived growth factor receptor beta phosphorylation in MG63 cells in the absence of plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50292533(CHEMBL446790 | Fukugetin)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50326050(CHEMBL1240617)
Affinity DataIC50:  3.40E+3nMAssay Description:Binding affinity to human kallikrein 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed