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Found 60 Enz. Inhib. hit(s) with Target = 'Promotilin'
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86314(CAS_0 | NSC_0 | [Nle13]-Motilin)
Affinity DataKi:  0.447nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86314(CAS_0 | NSC_0 | [Nle13]-Motilin)
Affinity DataKi:  0.850nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85994([leu13]pMOT(1-19))
Affinity DataKi:  0.980nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  0.980nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85614([Leu13]motilin | [leu13]pMOT(1-22))
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85614([Leu13]motilin | [leu13]pMOT(1-22))
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  1.29nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85979([ala3,leu13]pMOT(1-14))
Affinity DataKi:  1.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50143037(CHEMBL411576 | MOTILIN)
Affinity DataKi:  1.35nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86314(CAS_0 | NSC_0 | [Nle13]-Motilin)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86314(CAS_0 | NSC_0 | [Nle13]-Motilin)
Affinity DataKi:  1.95nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85987([leu13]pMOT(1-16))
Affinity DataKi:  2.14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85389(CAS_52906-92-0 | Motilin)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85389(CAS_52906-92-0 | Motilin)
Affinity DataKi:  2.82nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85389(CAS_52906-92-0 | Motilin)
Affinity DataKi:  3.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85981([ala1,leu13]pMOT(1-14) | [leu13]pMOT(1-14))
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85615(L-Phe-L-Val-L-Pro-L-Ile-L-Phe-L-Thr-L-Tyr-Gly-L-Gl...)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85615(L-Phe-L-Val-L-Pro-L-Ile-L-Phe-L-Thr-L-Tyr-Gly-L-Gl...)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85614([Leu13]motilin | [leu13]pMOT(1-22))
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85389(CAS_52906-92-0 | Motilin)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85986([ala11,leu13]pMOT(1-14))
Affinity DataKi:  4.57nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85992([ala10,leu13]pMOT(1-14))
Affinity DataKi:  5.01nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85389(CAS_52906-92-0 | Motilin)
Affinity DataKi:  5.25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85989(N-ethyl, N-methyl Erythromycin-A enol ether)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85980([ala12,leu13]pMOT(1-14))
Affinity DataKi:  6.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85999([ala14,leu13]pMOT(1-14))
Affinity DataKi:  7.08nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85990([ala13,leu13]pMOT(1-14))
Affinity DataKi:  7.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85993(Erythromycin-B enol ether)
Affinity DataKi:  7.59nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85846(CAS_33396-29-1 | EM523 | Erythromycin A 6,9-enolet...)
Affinity DataKi:  8.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85846(CAS_33396-29-1 | EM523 | Erythromycin A 6,9-enolet...)
Affinity DataKi:  19.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85984([ala5,leu13]pMOT(1-14))
Affinity DataKi:  28.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85390(GM 611 | Mitemcinal)
Affinity DataKi:  31.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85983([ala8,leu13]pMOT(1-14))
Affinity DataKi:  36.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85978([ala6,leu13]pMOT(1-14))
Affinity DataKi:  46.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85846(CAS_33396-29-1 | EM523 | Erythromycin A 6,9-enolet...)
Affinity DataKi:  47.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86675(CAS_0 | NSC_0 | [Bpa5,Ile13]Motilin | [L-Bpa5,Ile1...)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86675(CAS_0 | NSC_0 | [Bpa5,Ile13]Motilin | [L-Bpa5,Ile1...)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86685(ABT-229)
Affinity DataKi:  58.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85991([ala9,leu13]pMOT(1-14))
Affinity DataKi:  75.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85995([leu13]pMOT(1-11))
Affinity DataKi:  89.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85998(Erythromycin-B)
Affinity DataKi:  145nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(RABBIT)
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86313(CAS_114-07-8 | NSC_12560 | erythromycin-A)
Affinity DataKi:  191nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85988(N-ethyl, N-Methyl Erythromycin-A)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM85846(CAS_33396-29-1 | EM523 | Erythromycin A 6,9-enolet...)
Affinity DataKi:  257nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86688(EM-B enolether)
Affinity DataKi:  324nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86676([D-Bpa5,Ile13]Motilin)
Affinity DataKi:  420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86313(CAS_114-07-8 | NSC_12560 | erythromycin-A)
Affinity DataKi:  513nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Glaxosmithkline

Curated by PDSP Ki Database
LigandPNGBDBM86686(Erythromycin A Enol Ether | ME4)
Affinity DataKi:  537nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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