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Found 6 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-6/beta-4'
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50516340(CHEMBL4439678)
Affinity DataIC50:  17nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567426(CHEMBL4878856)
Affinity DataIC50:  23nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50567413(CHEMBL4865365)
Affinity DataIC50:  27nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50516342(CHEMBL4461998)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50445326(CHEMBL3104239)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-6/beta-4(Rattus norvegicus (Rat))
Veterans Affairs Medical Center

Curated by ChEMBL
LigandPNGBDBM50445326(CHEMBL3104239)
Affinity DataIC50:  222nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed